Synthesis and biological evaluation of new dipyrrolo[3,4-a:3,4-c]carbazole-1,3,4,6-tetraones, substituted with various saturated and unsaturated side chains via palladium catalyzed cross-coupling reactions.

نویسندگان

  • Hélène Hénon
  • Fabrice Anizon
  • Roy M Golsteyn
  • Stéphane Léonce
  • Robert Hofmann
  • Bruno Pfeiffer
  • Michelle Prudhomme
چکیده

The syntheses of a series of dipyrrolo[3,4-a:3,4-c]carbazole-1,3,4,6-tetraones, substituted in 10-position with saturated and unsaturated side chains, via palladium catalyzed cross-coupling reactions, are described. These compounds can be considered as granulatimide bis-imide analogues. Their inhibitory activity toward Chk1 kinase and their antiproliferative activities in vitro in four tumor cell lines are reported.

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عنوان ژورنال:
  • Bioorganic & medicinal chemistry

دوره 14 11  شماره 

صفحات  -

تاریخ انتشار 2006